BDBM35667 AVP::CHEMBL373742::US10131692, 44 (AVP)::[3H]Arginine vasopressin::[3H]Argipressin tannate::[3H]vasopressin
SMILES [#7]-[#6@H]-1-[#6]-[#16]-[#16]-[#6]-[#6@H](-[#7]-[#6](=O)-[#6@H](-[#6]-[#6](-[#7])=O)-[#7]-[#6](=O)-[#6@H](-[#6]-[#6]-[#6](-[#7])=O)-[#7]-[#6](=O)-[#6@H](-[#6]-c2ccccc2)-[#7]-[#6](=O)-[#6@H](-[#6]-c2ccc(-[#8])cc2)-[#7]-[#6]-1=O)-[#6](=O)-[#7]-1-[#6]-[#6]-[#6]-[#6@H]-1-[#6](=O)-[#7]-[#6@@H](-[#6]-[#6]-[#6]\[#7]=[#6](\[#7])-[#7])-[#6](=O)-[#7]-[#6]-[#6](-[#7])=O
InChI Key InChIKey=KBZOIRJILGZLEJ-LGYYRGKSSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 35667
Affinity DataEC50: 8.30nMAssay Description:Agonist activity at human oxytocin receptor expressed CHO cells assessed as induction of phospholipase C activity after 15 mins by inositol phosphate...More data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Agonist activity at human OT receptor expressed in CHO-K1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
Affinity DataEC50: 15nMAssay Description:Agonist activity at human OT receptor expressed in CHO-K1 cells by luciferase reporter gene assayMore data for this Ligand-Target Pair
TargetVasopressin V2 receptor(Homo sapiens (Human))
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Second Tokushima Institute of New Drug Research
Curated by PDSP Ki Database
Affinity DataEC50: 40nMAssay Description:Agonist activity of compounds on the human V2 receptor (h V2R) was determined in a transcriptional reporter gene assay by transiently transfecting an...More data for this Ligand-Target Pair
Affinity DataEC50: 5.40E+3nMAssay Description:To determine selectivity, compounds were tested in luciferase-based transcriptional reporter gene assays expressing the human V1b receptor (hV1bR). A...More data for this Ligand-Target Pair