BDBM383242 9-(4-chlorobenzyl)-6-methyl- 4-(2-((1-methyl-1H-pyrazol- 5-yl)amino)pyrimidin-4-yl)- 8,9-dihydro-1,2,2a1,6- tetraazabenzo[cd]azulen- 7(6H)-one::US10278975, Compound I-22 S::US11376260, Example I-22S
SMILES CN1c2cc(cc3nnc([C@@H](Cc4ccc(Cl)cc4)CC1=O)n23)-c1ccnc(Nc2ccnn2C)n1
InChI Key InChIKey=CLXYQKJFFSNBSK-KRWDZBQOSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 383242
Affinity DataIC50: <0.0200nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: <0.0200nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair