BDBM383314 4-(9-(4-fluorophenoxy)- 8,9-dihydro-7H-6-oxa- 1,2,2a1- triazabenzo[cd]azulen-4- yl)-N-(1-methyl-1H- pyrazol-5-yl)pyrimidin-2- amine::US10278975, Compound I-108 S::US10278975, Compound I-66 S::US11376260, Example I-108S
SMILES Cn1nccc1Nc1nccc(n1)-c1cc2OCC[C@H](Oc3ccc(F)cc3)c3nnc(c1)n23
InChI Key InChIKey=CTWHMTCAEZFXMK-SFHVURJKSA-N
Data 4 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 383314
Affinity DataIC50: 0.0200nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: <0.0200nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: 0.0200nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: <0.0200nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair