BDBM383361 N-(1-methyl-1H-pyrazol-5- yl)-4-(9-((3-methylisoxazol- 5-yl)methyl)-8,9-dihydro-7H- 6-oxa-1,2,2a1- triazabenzo[cd]azulen-4- yl)pyrimidin-2-amine::US10278975, Compound I-93 S::US11376260, Example I-93R
SMILES Cc1cc(C[C@H]2CCOc3cc(cc4nnc2n34)-c2ccnc(Nc3ccnn3C)n2)on1
InChI Key InChIKey=VPKQELJVDUHMBF-CQSZACIVSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 383361
Affinity DataIC50: <0.0200nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair
Affinity DataIC50: 18.2nMAssay Description:Compounds were tested in an enzymatic assay using human ERK-2 (Mitogen Activated Kinase 1), recombinantly expressed as an n-terminal 6-His fusion pro...More data for this Ligand-Target Pair