BDBM4117 3-phenyl-1-(1,2,6,7-tetrahydroxy-9H-carbazol-9-yl)propan-1-one::Carbazole deriv. 9aa

SMILES Oc1ccc2c3cc(O)c(O)cc3n(C(=O)CCc3ccccc3)c2c1O

InChI Key InChIKey=RCNJNRIRPVQSJH-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 4117   

LigandPNGBDBM4117(3-phenyl-1-(1,2,6,7-tetrahydroxy-9H-carbazol-9-yl)...)
Affinity DataIC50:  2.30E+3nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of PKA activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] label...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Pfizer

LigandPNGBDBM4117(3-phenyl-1-(1,2,6,7-tetrahydroxy-9H-carbazol-9-yl)...)
Affinity DataIC50:  400nMAssay Description:IC50 is the inhibitor concentration, which inhibits 50% of pp60c-src activity that catalyzes the transfer of the terminal phosphate from [gamma-32P] ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed