BDBM453212 1-(5-fluoro-2-methoxy-4-(((1R,2R)-2- (trifluoromethyl)cyclopropyl)ethynyl)phenyl)-N-3- isoxazolyl-2-oxo-1,2-dihydro-6-quinolinesulfonamide::US10729684, Example 5
SMILES COc1cc(C#CC2(CC2)C(F)(F)F)c(F)cc1-n1c2ccc(cc2ccc1=O)S(=O)(=O)Nc1ccon1
InChI Key InChIKey=UMIDIJOAHPZCQY-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 453212
Affinity DataIC50: 62nMAssay Description:HEK 293 cells stably transfected with human Nav1.7 were recorded in whole cell voltage clamp mode with the PatchXpress automated electrophysiology sy...More data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:HEK 293 Cells stably transfected with either Nav 1.7 or Nav 1.5 were recorded in population patch-clamp mode with the IonWorks® Quattro automated ele...More data for this Ligand-Target Pair