BDBM50000296 CHEMBL441765::CHEMBL482811::U-50488H::US11492374, ID 1
SMILES CN([C@@H]1CCCC[C@H]1N1CCCC1)C(=O)Cc1ccc(Cl)c(Cl)c1
InChI Key InChIKey=VQLPLYSROCPWFF-QZTJIDSGSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50000296
Affinity DataKi: 0.600nMAssay Description:Displacement of [3H]U69593 from rat KOR expressed in CHO cellsMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Catania
Curated by ChEMBL
University Of Catania
Curated by ChEMBL
Affinity DataKi: 1.10nMAssay Description:Displacement of [3H]U69593 from Sprague-Dawley rat kappa opioid receptor in guinea pig cerebella by liquid scintillation countingMore data for this Ligand-Target Pair
TargetKappa-type opioid receptor(Cavia porcellus (domestic guinea pig))
University Of Catania
Curated by ChEMBL
University Of Catania
Curated by ChEMBL
Affinity DataKi: 5nMAssay Description:Displacement of [3H]-U-69,593 from Opioid receptor kappa 1 in guinea pig cerebellar.More data for this Ligand-Target Pair
Affinity DataKi: 716nMAssay Description:Tested for binding affinity by [3H]diprenorphine displacement for Opioid receptor mu 1 was carried on crude membrane fractions obtained from the whol...More data for this Ligand-Target Pair
Affinity DataKi: 1.75E+3nMAssay Description:Displacement of [3H]DAMGO from Sprague-Dawley rat mu opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: >5.00E+3nMAssay Description:Displacement of [3H]DPDPE from Sprague-Dawley rat delta opioid receptor by liquid scintillation countingMore data for this Ligand-Target Pair
Affinity DataKi: 8.10E+3nMAssay Description:Tested for binding affinity by [3H]diprenorphine displacement for Opioid receptor delta 1 are carried on crude membrane fractions obtained from the w...More data for this Ligand-Target Pair