BDBM50005917 CHEMBL3234681

SMILES [H][C@]12CC[C@]([H])(C1)c1c2c(nn1-c1ccc(F)cc1F)C(=O)NC(C)(C)C

InChI Key InChIKey=NTPZXHMTJGOMCJ-WDEREUQCSA-N

Data  3 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50005917   

TargetCannabinoid receptor 2(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50005917(CHEMBL3234681)
Affinity DataKi:  12nMAssay Description:Agonist activity at human CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Rattus norvegicus (Rat))
Arena Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50005917(CHEMBL3234681)
Affinity DataKi:  12nMAssay Description:Binding affinity to rat CB2 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50005917(CHEMBL3234681)
Affinity DataKi:  985nMAssay Description:Agonist activity at human CB1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50005917(CHEMBL3234681)
Affinity DataEC50:  0.610nMAssay Description:Agonist activity at human CB2 receptor assessed as inhibition of forskolin-induced cAMP production preincubated for 15 mins followed by forskolin cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Univ. Lille

Curated by ChEMBL
LigandPNGBDBM50005917(CHEMBL3234681)
Affinity DataEC50:  854nMAssay Description:Agonist activity at human CB1 receptor assessed as inhibition of forskolin-induced cAMP production preincubated for 15 mins followed by forskolin cha...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed