BDBM50007428 7-[3-(4-Pyridin-2-yl-piperazin-1-yl)-propoxy]-chromen-4-one::CHEMBL84639
SMILES O=c1ccoc2cc(OCCCN3CCN(CC3)c3ccccn3)ccc12
InChI Key InChIKey=NVGYZBZAFVGARK-UHFFFAOYSA-N
Data 7 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50007428
Affinity DataIC50: 2.17E+4nMAssay Description:Compound was tested for its inhibitory effect on the binding profile in Dopamine receptor D1 using [3H]flupenthixol in rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 1.08E+3nMAssay Description:Compound was tested for its inhibitory effect on the binding profile in Dopamine receptor D2 using [3H]haloperidol in rat brain.More data for this Ligand-Target Pair
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was tested for its inhibitory effect on the binding profile in 5-hydroxytryptamine 2 receptor using [3H]spiroperidol in rat brain.More data for this Ligand-Target Pair
TargetAlpha-1A/Alpha-1B/Alpha-1D adrenergic receptor(Rattus norvegicus (rat))
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 170nMAssay Description:Compound was tested for its inhibitory effect on the binding profile in Alpha-1 adrenergic receptor using [3H]prazosin in rat brain.More data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 59nMAssay Description:Compound was tested for its inhibitory effect on the binding profile in Dopamine receptor using [3H]N-propylnorapomorphine in rat brain.More data for this Ligand-Target Pair
TargetAlpha-2A adrenergic receptor [16-465]/Alpha-2B adrenergic receptor/Alpha-2C adrenergic receptor(RAT)
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 2.60E+3nMAssay Description:Compound was tested for its inhibitory effect on the binding profile in Alpha-2 adrenergic receptor using [3H]p-aminoclonidine in rat brain.More data for this Ligand-Target Pair
TargetD(1A)/D(1B)/D(2)/D(3)/D(4) dopamine receptor(Rattus norvegicus (rat))
Warner-Lambert
Curated by ChEMBL
Warner-Lambert
Curated by ChEMBL
Affinity DataIC50: 1.00E+3nMAssay Description:Compound was tested for inhibitory binding activity against Dopamine receptor in rat striatal membranes using [3H]HAL as the radioligand.More data for this Ligand-Target Pair