BDBM50034993 (S)-6-Amino-2-[(S)-3-hydroxy-2-(2-{4-[4-(2-methyl-imidazol-1-yl)-butyl]-phenyl}-acetylamino)-propionylamino]-hexanoic acid (2-cyclohexyl-ethyl)-amide::CHEMBL6269::SC-58272::[CYCLOHEXYLETHYL]-[[[[4-[2-METHYL-1-IMIDAZOLYL-BUTYL]PHENYL]ACETYL]-SERYL]-LYSINYL]-AMINE
SMILES Cc1nccn1CCCCc1ccc(CC(=O)N[C@@H](CO)C(=O)N[C@@H](CCCCN)C(=O)NCCC2CCCCC2)cc1
InChI Key InChIKey=WHLPIOSHBKQGHA-KYJUHHDHSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 12 hits for monomerid = 50034993
TargetGlycylpeptide N-tetradecanoyltransferase(Candida albicans (Yeast))
G.D. Searle And
Curated by ChEMBL
G.D. Searle And
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:The Compound was tested for the inhibition potency against C. albicans N-myristoyltransferase (NMT) and reported as apparent KiMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1/2(Homo sapiens (Human))
G.D. Searle And
Curated by ChEMBL
G.D. Searle And
Curated by ChEMBL
Affinity DataKi: 31nMAssay Description:Apparent binding affinity against Candida albicans N-Myristoyltransferase (NMT).More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1/2(Homo sapiens (Human))
G.D. Searle And
Curated by ChEMBL
G.D. Searle And
Curated by ChEMBL
Affinity DataIC50: >1.40E+5nMAssay Description:Inhibitory activity against human N-myristoyltransferase (HsNmt)More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase(Saccharomyces cerevisiae)
Chinese Academy Of Sciences
Curated by ChEMBL
Chinese Academy Of Sciences
Curated by ChEMBL
Affinity DataIC50: 24nMAssay Description:Inhibition of Saccharomyces cerevisiae NMTMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1/2(Homo sapiens (Human))
G.D. Searle And
Curated by ChEMBL
G.D. Searle And
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition of Candida albicans N-myristoyltransferase (NMT) with peptide GNAASARR-NH2 and [3H]myristoyl-CoA at 1 uMMore data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1/2(Homo sapiens (Human))
G.D. Searle And
Curated by ChEMBL
G.D. Searle And
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibition activity against N-myristoyltransferase (NMT) of candida albicans.More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1/2(Homo sapiens (Human))
G.D. Searle And
Curated by ChEMBL
G.D. Searle And
Curated by ChEMBL
Affinity DataIC50: 1.41E+4nMAssay Description:Inhibition activity against N-myristoyltransferase (NMT) of human.More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1/2(Homo sapiens (Human))
G.D. Searle And
Curated by ChEMBL
G.D. Searle And
Curated by ChEMBL
Affinity DataIC50: 1.41E+4nMAssay Description:Inhibitory activity against human N-Myristoyltransferase (NMT).More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1/2(Homo sapiens (Human))
G.D. Searle And
Curated by ChEMBL
G.D. Searle And
Curated by ChEMBL
Affinity DataIC50: 56nMAssay Description:Inhibitory activity against Candida albicans N-Myristoyltransferase (NMT).More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1/2(Homo sapiens (Human))
G.D. Searle And
Curated by ChEMBL
G.D. Searle And
Curated by ChEMBL
Affinity DataIC50: 830nMAssay Description:Inhibitory activity against Candida albicans N-myristoyltransferase (CaNmt)More data for this Ligand-Target Pair
Affinity DataIC50: 60nMAssay Description:Compound was tested for its inhibitory activity against Candida albicans N-Myristoyltransferase (NMT)More data for this Ligand-Target Pair
TargetGlycylpeptide N-tetradecanoyltransferase 1/2(Homo sapiens (Human))
G.D. Searle And
Curated by ChEMBL
G.D. Searle And
Curated by ChEMBL
Affinity DataIC50: 1.41E+4nMAssay Description:Tested for Inhibitory concentration against human N-myristoyltransferase (NMT) in radiochemical HPLC end point assay with peptide GNAASARR-NH2 and [3...More data for this Ligand-Target Pair