BDBM50036705 CHEMBL3354816

SMILES CN[C@@H]1CCN(C1)c1ccnc(NC(C)C)c1

InChI Key InChIKey=BVMYJSFGALTWOF-LLVKDONJSA-N

Data  2 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50036705   

TargetHistamine H4 receptor(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50036705(CHEMBL3354816)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]histamine from human recombinant histamine H4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50036705(CHEMBL3354816)
Affinity DataKi:  19nMAssay Description:Displacement of [3H]histamine from human recombinant histamine H4 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H4 receptor(Homo sapiens (Human))
Janssen Research And Development

Curated by ChEMBL
LigandPNGBDBM50036705(CHEMBL3354816)
Affinity DataEC50:  3.16E+3nMAssay Description:Agonist activity at human recombinant histamine H4 receptor expressed in SK-N-MC cells assessed as effect on forskolin-stimulated cAMP-mediated repor...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed