BDBM50056420 4-Amino-5-chloro-2-methoxy-benzoic acid 2-(4-benzoyl-piperidin-1-yl)-ethyl ester::CHEMBL160237
SMILES COc1cc(N)c(Cl)cc1C(=O)OCCN1CCC(CC1)C(=O)c1ccccc1
InChI Key InChIKey=NCJGDEWUYHFOFK-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 50056420
Affinity DataKi: 7.60nMAssay Description:Binding affinity towards 5-hydroxytryptamine 4 receptor was determined in rat striatal membranes using [3H]GR-113808 as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 100nMAssay Description:5-hydroxytryptamine 4 receptor antagonist activity, concentration which gave 50% reduction of the 5-HT-induced contractions in the guinea pig ileumMore data for this Ligand-Target Pair