BDBM50074997 (E)-3-(6-Acetylamino-pyridin-3-yl)-N-({[4-methoxy-3-(2-methyl-quinolin-8-yloxymethyl)-2-methylsulfanyl-phenyl]-methyl-carbamoyl}-methyl)-acrylamide::CHEMBL115163
SMILES COc1ccc(N(C)C(=O)CNC(=O)\C=C\c2ccc(NC(C)=O)nc2)c(SC)c1COc1cccc2ccc(C)nc12
InChI Key InChIKey=LQLXUORFZSRSRP-LFIBNONCSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 50074997
Affinity DataKi: 0.600nMAssay Description:Inhibition of BK-induced (4x10E-8M) contraction of isolated guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataIC50: 5.20nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair
Affinity DataEC50: 59nMAssay Description:Inhibition of specific binding of [3H]-BK to bradykinin B2 receptors of guinea pig ileum (GPI)More data for this Ligand-Target Pair