BDBM50089958 CHEMBL3581226

SMILES CC(C)(C)c1cc(cc(c1O)C(C)(C)C)-c1csc(n1)C1(CCOCC1)N1CCCCC1

InChI Key InChIKey=COLTZBDSWGVCQJ-UHFFFAOYSA-N

Data  2 KI  2 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50089958   

TargetCannabinoid receptor 2(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089958(CHEMBL3581226)
Affinity DataKi:  50nMAssay Description:Displacement of [3H]CP55940 from human CB2 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089958(CHEMBL3581226)
Affinity DataKi:  2.17E+3nMAssay Description:Displacement of [3H]CP55940 from human CB1 receptor expressed in CHO-K1 cell membrane by competitive displacement assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089958(CHEMBL3581226)
Affinity DataEC50:  40nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Ipsen Innovation

Curated by ChEMBL
LigandPNGBDBM50089958(CHEMBL3581226)
Affinity DataEC50:  2.26E+3nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO-K1 cells assessed as inhibition of forskolin-stimulated cAMP productionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed