BDBM50109544 3-[4-(2-beta-Carbolin-9-yl-ethoxy)-phenyl]-2-ethoxy-propionic acid::CHEMBL166637

SMILES CCO[C@@H](Cc1ccc(OCCn2c3ccccc3c3ccncc23)cc1)C(O)=O

InChI Key InChIKey=OCSNIPAKIFPWTJ-QHCPKHFHSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50109544   

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50109544(3-[4-(2-beta-Carbolin-9-yl-ethoxy)-phenyl]-2-ethox...)
Affinity DataEC50:  11nMAssay Description:In vitro transactivation using receptor transactivation assay against hPPAR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Novo Nordisk

Curated by ChEMBL
LigandPNGBDBM50109544(3-[4-(2-beta-Carbolin-9-yl-ethoxy)-phenyl]-2-ethox...)
Affinity DataEC50:  11nMAssay Description:Transactivation of Homo sapiens (human) PPARgamma assessed as luciferase activity by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50109544(3-[4-(2-beta-Carbolin-9-yl-ethoxy)-phenyl]-2-ethox...)
Affinity DataEC50:  141nMAssay Description:Transactivation of Homo sapiens (human) PPARalpha assessed as luciferase activity by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50109544(3-[4-(2-beta-Carbolin-9-yl-ethoxy)-phenyl]-2-ethox...)
Affinity DataEC50:  140nMAssay Description:In vitro transactivation using receptor transactivation assay against hPPAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed