BDBM50126544 4-(5-{[{4-[4-(5-Chloro-thiophene-2-carbonyl)-piperazin-1-yl]-phenyl}-(4-fluoro-benzyl)-amino]-methyl}-imidazol-1-ylmethyl)-benzonitrile::CHEMBL36529

SMILES Fc1ccc(CN(Cc2cncn2Cc2ccc(cc2)C#N)c2ccc(cc2)N2CCN(CC2)C(=O)c2ccc(Cl)s2)cc1

InChI Key InChIKey=MDOLNMYVGZJXLJ-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50126544   

TargetProtein farnesyltransferase subunit beta/geranylgeranyltransferase type-1 subunit alpha(Bos taurus (bovine))
Centre De Recherche Pierre Fabre

Curated by ChEMBL
LigandPNGBDBM50126544(4-(5-{[{4-[4-(5-Chloro-thiophene-2-carbonyl)-piper...)
Affinity DataIC50:  70nMAssay Description:Inhibit of purified bovine Farnesyl protein transferase.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed