BDBM50158041 1-Benzenesulfonyl-3-(1,2,3,6-tetrahydro-pyridin-4-yl)-1H-indole::CHEMBL179592

SMILES O=S(=O)(c1ccccc1)n1cc(C2=CCNCC2)c2ccccc12

InChI Key InChIKey=GOCDLKCFBOWAOO-UHFFFAOYSA-N

Data  2 KI  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50158041   

Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50158041(1-Benzenesulfonyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataKi:  2nMAssay Description:Binding affinity against cloned human 5-hydroxytryptamine 6 receptor expressed in HeLa cells using [3H]-LSDMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50158041(1-Benzenesulfonyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataKi:  2nMAssay Description:Displacement of [3H]-LSD from cloned human 5-hydroxytryptamine 6 receptor expressed in HeLa cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
Target5-hydroxytryptamine receptor 6(Homo sapiens (Human))
Wyeth Research

Curated by ChEMBL
LigandPNGBDBM50158041(1-Benzenesulfonyl-3-(1,2,3,6-tetrahydro-pyridin-4-...)
Affinity DataIC50:  43nMAssay Description:Inhibitory concentration against 5-HT stimulated cAMP production in HeLa cells stably transfected with human 5-HT6 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed