BDBM50179246 2-{4-[3-(2-phenyl-7-propyl-1H-indol-6-yloxy)propoxy]-indol-1-yl}ethanoic acid::CHEMBL198786

SMILES CCCc1c(OCCCOc2cccc3n(CC(O)=O)ccc23)ccc2cc([nH]c12)-c1ccccc1

InChI Key InChIKey=YRFJWRCVNFMVHJ-UHFFFAOYSA-N

Data  1 IC50  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50179246   

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179246(2-{4-[3-(2-phenyl-7-propyl-1H-indol-6-yloxy)propox...)
Affinity DataIC50:  1.68E+3nMAssay Description:Displacement of [3H]-rosiglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179246(2-{4-[3-(2-phenyl-7-propyl-1H-indol-6-yloxy)propox...)
Affinity DataEC50:  2.82E+3nMAssay Description:Functional activity at human PPAR gamma in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179246(2-{4-[3-(2-phenyl-7-propyl-1H-indol-6-yloxy)propox...)
Affinity DataEC50:  3.34E+3nMAssay Description:Functional activity at human PPAR delta in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
National Health Research Institutes

Curated by ChEMBL
LigandPNGBDBM50179246(2-{4-[3-(2-phenyl-7-propyl-1H-indol-6-yloxy)propox...)
Affinity DataEC50:  500nMAssay Description:Functional activity at human PPAR alpha in Huh7 cells by transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed