BDBM50188028 2-ethoxy-3-(1-((5-methyl-2-o-tolyloxazol-4-yl)methyl)-1H-indol-5-yl)propanoic acid::CHEMBL211371

SMILES CCOC(Cc1ccc2n(Cc3nc(oc3C)-c3ccccc3C)ccc2c1)C(O)=O

InChI Key InChIKey=QWORIWQTCIYNKN-UHFFFAOYSA-N

Data  2 IC50  3 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50188028   

TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50188028(2-ethoxy-3-(1-((5-methyl-2-o-tolyloxazol-4-yl)meth...)
Affinity DataEC50:  990nMAssay Description:Activity at PPARgamma by luciferase reporter gene transactivation assay relative to edaglitazoneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor delta(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50188028(2-ethoxy-3-(1-((5-methyl-2-o-tolyloxazol-4-yl)meth...)
Affinity DataEC50:  6.50E+3nMAssay Description:Activity at PPARdelta by luciferase reporter gene transactivation assay relative to GW 501516More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50188028(2-ethoxy-3-(1-((5-methyl-2-o-tolyloxazol-4-yl)meth...)
Affinity DataIC50:  125nMAssay Description:Binding affinity to PPARalpha by radio ligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50188028(2-ethoxy-3-(1-((5-methyl-2-o-tolyloxazol-4-yl)meth...)
Affinity DataIC50:  316nMAssay Description:Binding affinity to PPARgamma by radio ligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50188028(2-ethoxy-3-(1-((5-methyl-2-o-tolyloxazol-4-yl)meth...)
Affinity DataEC50:  830nMAssay Description:Activity at PPARalpha by luciferase reporter gene transactivation assay relative to farglitazarMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed