BDBM50190657 CHEMBL1194747
SMILES [H][C@@]12C[C@@]34[C@@H](O)[C@@]([H])(C(=O)C=C3S1)[N+]1=C3c5c(CC1)c[nH]c5C(=O)C(N2)=C43
InChI Key InChIKey=QJMJSLBHDYZDDN-JRXCTEAYSA-O
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50190657
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Maribor
Curated by ChEMBL
University Of Maribor
Curated by ChEMBL
Affinity DataKi: 1.50E+4nMAssay Description:Reversible competitive inhibition of electric eel AChE using acetylthiocholine iodide as substrate measured over 5 mins by Dixon plot analysisMore data for this Ligand-Target Pair
Affinity DataIC50: 5.31E+5nMAssay Description:Histamine H2 receptor antagonistic activity at a concentration of 1 uM on the isolated guinea pig right atrium.More data for this Ligand-Target Pair
Affinity DataIC50: 1.58E+5nMAssay Description:Inhibition of human AChE using acetylthiocholine iodide as substrate measured over 5 mins by Ellman's methodMore data for this Ligand-Target Pair
TargetHypoxia-inducible factor 1-alpha(Homo sapiens (Human))
National Cancer Institute-Frederick
Curated by ChEMBL
National Cancer Institute-Frederick
Curated by ChEMBL
Affinity DataIC50: 730nMAssay Description:Displacement of GST-tagged p300-CH1 domain (323 to 423 residues) from synthetic biotinylated HIF-1alpha C-TAD domain (786 to 826 residues) (unknown o...More data for this Ligand-Target Pair
TargetAcetylcholinesterase(Electrophorus electricus (Electric eel))
University Of Maribor
Curated by ChEMBL
University Of Maribor
Curated by ChEMBL
Affinity DataIC50: 2.57E+4nMAssay Description:Binding activity against Endothelin A receptor of Porcine aortic smooth muscle membranesMore data for this Ligand-Target Pair