BDBM50200356 Ac-c[Cys-His-D-Phe-Cys]-N-alpha-guanidinylbutyl-D-Trp-NH2::CHEMBL384955

SMILES CC(=O)N[C@H]1CSSC[C@H](NC(=O)[C@@H](Cc2ccccc2)NC(=O)[C@H](Cc2cnc[nH]2)NC1=O)C(=O)N(CCCCN=C(N)N)[C@H](Cc1c[nH]c2ccccc12)C(N)=O

InChI Key InChIKey=ZAKACLKQLDVSMU-ISBPOBPSSA-N

Data  2 IC50  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50200356   

TargetMelanocortin receptor 3(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50200356(Ac-c[Cys-His-D-Phe-Cys]-N-alpha-guanidinylbutyl-D-...)
Affinity DataIC50: >1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC3 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50200356(Ac-c[Cys-His-D-Phe-Cys]-N-alpha-guanidinylbutyl-D-...)
Affinity DataEC50: >1.00E+3nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMelanocortin receptor 4(Homo sapiens (Human))
University Of Arizona

Curated by ChEMBL
LigandPNGBDBM50200356(Ac-c[Cys-His-D-Phe-Cys]-N-alpha-guanidinylbutyl-D-...)
Affinity DataIC50:  0.700nMAssay Description:Displacement of [125I]NDP-alphaMSH from human MC4 receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed