BDBM50220703 (R)-N-((S)-3-(4-chlorophenyl)-1-(4-cyclohexyl-4-((1-methyl-1H-tetrazol-5-yl)methyl)piperidin-1-yl)-1-oxopropan-2-yl)-1,2,3,4-tetrahydroisoquinoline-3-carboxamide::CHEMBL250508
SMILES Cn1nnnc1CC1(CCN(CC1)C(=O)[C@H](Cc1ccc(Cl)cc1)NC(=O)[C@H]1Cc2ccccc2CN1)C1CCCCC1
InChI Key InChIKey=IJYUZXAPJHBRJR-WDYNHAJCSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50220703
Affinity DataEC50: 115nMAssay Description:Antagonist activity at human MC3R assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataIC50: 0.850nMAssay Description:Binding affinity to human MC4RMore data for this Ligand-Target Pair
Affinity DataEC50: 222nMAssay Description:Antagonist activity at human MC5R assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair
Affinity DataEC50: 3.20nMAssay Description:Antagonist activity at human MC4R assessed as stimulation of cAMP productionMore data for this Ligand-Target Pair