BDBM50254144 2-(4-chlorophenylsulfonyl)-2-methyl-N-(5-(5-methylthiophen-2-yl)pyridin-3-yl)propanamide::CHEMBL466821

SMILES Cc1ccc(s1)-c1cncc(NC(=O)C(C)(C)S(=O)(=O)c2ccc(Cl)cc2)c1

InChI Key InChIKey=SELHIMASMNUSIZ-UHFFFAOYSA-N

Data  4 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50254144   

TargetCannabinoid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50254144(2-(4-chlorophenylsulfonyl)-2-methyl-N-(5-(5-methyl...)
Affinity DataEC50:  9nMAssay Description:Agonist activity at human CB2 receptor expressed in SF9 cells assessed as inhibition of CP55940-stimulated GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50254144(2-(4-chlorophenylsulfonyl)-2-methyl-N-(5-(5-methyl...)
Affinity DataEC50:  322nMAssay Description:Agonist activity at human CB1 receptor expressed in SF9 cells assessed as inhibition of CP55940-stimulated GTP bindingMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 1(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50254144(2-(4-chlorophenylsulfonyl)-2-methyl-N-(5-(5-methyl...)
Affinity DataEC50:  331nMAssay Description:Agonist activity at human CB1 receptor expressed in CHO cells assessed as suppression of forskolin-stimulated cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetCannabinoid receptor 2(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50254144(2-(4-chlorophenylsulfonyl)-2-methyl-N-(5-(5-methyl...)
Affinity DataEC50:  5nMAssay Description:Agonist activity at human CB2 receptor expressed in CHO cells assessed as suppression of forskolin-stimulated cAMP accumulationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed