BDBM50257034 CHEMBL4096543
SMILES CC(C)Oc1cccnc1N(C)C1CCN(Cc2ccc(I)cc2)CC1
InChI Key InChIKey=ZJAXDNQQFMPNAV-UHFFFAOYSA-N
Data 11 KI
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 11 hits for monomerid = 50257034
TargetD(4) dopamine receptor(Homo sapiens (Human))
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:Inhibition of human dopamine D4 receptorMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataKi: 0.330nMAssay Description:Displacement of [3H]-spiperone from D4 (unknown origin) receptor expressed in CHO cells assessed as inhibition constantMore data for this Ligand-Target Pair
TargetD(4) dopamine receptor(Homo sapiens (Human))
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataKi: 0.331nMAssay Description:Displacement of [3H]N-methylspiperone from human dopamine D4 receptor expressed in HEK293 cell membranes after 1 hr by scintillation counting methodMore data for this Ligand-Target Pair
TargetSigma non-opioid intracellular receptor 1(Homo sapiens (Human))
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataKi: 82nMAssay Description:Inhibition of sigma1 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 145nMAssay Description:Displacement of [3H]-spiperone from human D3 receptor expressed in CCCL-1 cells assessed as inhibition constantMore data for this Ligand-Target Pair
TargetD(3) dopamine receptor(Homo sapiens (Human))
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataKi: 145nMAssay Description:Inhibition of human dopamine D3 receptorMore data for this Ligand-Target Pair
Target5-hydroxytryptamine receptor 2A(Homo sapiens (Human))
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataKi: 273nMAssay Description:Inhibition of serotonin 5-HT2 receptor (unknown origin)More data for this Ligand-Target Pair
Affinity DataKi: 568nMAssay Description:Displacement of [3H]-spiperone from human D2 receptor expressed in Sf9 cells assessed as inhibition constantMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+3nMAssay Description:Inhibition of human dopamine D2 (long) receptor (unknown origin)More data for this Ligand-Target Pair
TargetD(1A) dopamine receptor(Homo sapiens (Human))
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataKi: 2.83E+3nMAssay Description:Inhibition of human dopamine D1 receptorMore data for this Ligand-Target Pair
TargetD(1B) dopamine receptor(Homo sapiens (Human))
University of Nebraska Medical Center
Curated by ChEMBL
University of Nebraska Medical Center
Curated by ChEMBL
Affinity DataKi: >1.00E+4nMAssay Description:Inhibition of human dopamine D5 receptorMore data for this Ligand-Target Pair