BDBM50257992 (1S,3R)-N-(3,5-bis(trifluoromethyl)benzyl)-3-(2,3-dihydro-1H-inden-1-ylamino)-1-isopropylcyclopentanecarboxamide::CHEMBL494019
SMILES CC(C)[C@@]1(CC[C@H](C1)NC1CCc2ccccc12)C(=O)NCc1cc(cc(c1)C(F)(F)F)C(F)(F)F
InChI Key InChIKey=YYRQKVPZQIKPRY-KYPFDINASA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50257992
Affinity DataKi: 50nMAssay Description:Displacement of [125I]-CCL2 from human CCR2 receptor expressed in human U2OS cell membranesMore data for this Ligand-Target Pair
Affinity DataKi: 50nMAssay Description:Displacement of 0.1 nM [125I]CCL2 from human CCR2 expressing human U2OS cell membrane by scintillation spectrometryMore data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Antagonist activity at CCR2 (unknown origin)More data for this Ligand-Target Pair
Affinity DataIC50: 77nMAssay Description:Displacement of [125I]hMCP1 from human CCR2 receptor expressed in CHO cellsMore data for this Ligand-Target Pair