BDBM50263294 3-(4-{[3-(1-Azepanyl)propyl]oxy}phenyl)-2-methyl-4(3H)-quinazolinone::CHEMBL476579

SMILES Cc1nc2ccccc2c(=O)n1-c1ccc(OCCCN2CCCCCC2)cc1

InChI Key InChIKey=YJAKSFIWYQQJBZ-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50263294   

TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50263294(3-(4-{[3-(1-Azepanyl)propyl]oxy}phenyl)-2-methyl-4...)
Affinity DataIC50:  6.60E+3nMAssay Description:Displacement of [35S]N-[(4R)-1'-[(2R)-6-cyano-1,2,3,4-tetrahydro-2-naphthalenyl]-3,4-dihydro-4-hydroxyspiro[2H-1-benzopyran-2,4'-piperidin]-6-yl]meth...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Homo sapiens (Human))
Tsukuba Research Institute

Curated by ChEMBL
LigandPNGBDBM50263294(3-(4-{[3-(1-Azepanyl)propyl]oxy}phenyl)-2-methyl-4...)
Affinity DataIC50:  1.60nMAssay Description:Displacement of [3H]N-alpha-methylhistamine from human histamine H3 receptor expressed in CHO-K1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed