BDBM50264801 3-(2-chloro-6-fluorophenyl)-5-(2-(4-fluoropiperidin-4-yl)-1-methyl-1H-imidazol-5-yl)isoxazole::CHEMBL490430

SMILES Cn1c(cnc1C1(F)CCNCC1)-c1cc(no1)-c1c(F)cccc1Cl

InChI Key InChIKey=BQFJTJDULYXNJI-UHFFFAOYSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50264801   

TargetNeuronal acetylcholine receptor subunit alpha-4(Homo sapiens (Human))
Amgen

Curated by ChEMBL
LigandPNGBDBM50264801(3-(2-chloro-6-fluorophenyl)-5-(2-(4-fluoropiperidi...)
Affinity DataEC50:  34nMAssay Description:Activation of human alpha4beta2 nAChR assessed as potentiation of submaximal response to nicotine induced currentMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed