BDBM50269381 CHEMBL4100738

SMILES [H][C@@]12CC[C@@]([H])(C1)[C@H](C2)N1CCN(CC1)c1ccc(Nc2nc(N)n(n2)-c2nc(Cl)nc3c(C)csc23)cc1Cl

InChI Key InChIKey=VMMYOXWMJSIMQE-GUXCAODWSA-N

Data  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50269381   

TargetTyrosine-protein kinase receptor UFO(Homo sapiens (Human))
Rigel Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50269381(CHEMBL4100738)
Affinity DataEC50:  136nMAssay Description:Inhibition of Axl in human HeLa cells assessed as reduction in AKT phosphorylation at Ser 473 residues pre-incubated for 1 hr before preclustered ant...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed