BDBM50273469 CHEMBL4126406

SMILES [I-].Cc1oc2ccccc2c1C(=O)c1ccc(OCCC[N+](C)(C)C)cc1

InChI Key InChIKey=FKSGUSGEWAFUAT-UHFFFAOYSA-N

Data  6 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 6 hits for monomerid = 50273469   

TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50273469(CHEMBL4126406)
Affinity DataIC50:  1.26E+5nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7B (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase PHF2(Homo sapiens)
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50273469(CHEMBL4126406)
Affinity DataIC50:  5.98E+5nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7C (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistone lysine demethylase PHF8(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50273469(CHEMBL4126406)
Affinity DataIC50:  3.10E+5nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7B (PHD) (unknown origin) preincubated for 15 mins followed by p...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50273469(CHEMBL4126406)
Affinity DataIC50:  5.60E+3nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 7A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50273469(CHEMBL4126406)
Affinity DataIC50:  5.60E+3nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from KDM7A (PHD-JmjC) (unknown origin) preincubated for 15 mins followed...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetLysine-specific demethylase 5A(Homo sapiens (Human))
University Of Oxford

Curated by ChEMBL
LigandPNGBDBM50273469(CHEMBL4126406)
Affinity DataIC50:  8.44E+5nMAssay Description:Displacement of C-terminally biotinylated-H3K4me3 (1 to 21 residues) peptide from recombinant His6-tagged human KDM5A (PHD3) (1542 to 1660 residues) ...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed