BDBM50279103 5-(thiophen-2-ylsulfonyl)-5H-dibenzo[b,d]azepin-7(6H)-one::CHEMBL497249

SMILES O=C1CN(c2ccccc2-c2ccccc12)S(=O)(=O)c1cccs1

InChI Key InChIKey=YORIAFCWXUMHOS-UHFFFAOYSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50279103   

LigandPNGBDBM50279103(5-(thiophen-2-ylsulfonyl)-5H-dibenzo[b,d]azepin-7(...)
Affinity DataIC50:  2.40E+3nMAssay Description:Inhibition of human cloned IK1 expressed in african green monkey COS7 cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPotassium voltage-gated channel subfamily A member 3(Homo sapiens (Human))
4Sc

Curated by ChEMBL
LigandPNGBDBM50279103(5-(thiophen-2-ylsulfonyl)-5H-dibenzo[b,d]azepin-7(...)
Affinity DataIC50:  1.30E+4nMAssay Description:Inhibition of cloned Kv1.3 channel (unknown origin) expressed in mammalian cells by whole cell patch clamp assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed