BDBM50287161 4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2-(4-phenyl-piperazin-1-yl)-ethyl]-amide::CHEMBL30208

SMILES COc1c(cc(Br)c2ccccc12)C(=O)NCCN1CCN(CC1)c1ccccc1

InChI Key InChIKey=COCBRLNWXSGWJZ-UHFFFAOYSA-N

Data  3 KI  1 EC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 4 hits for monomerid = 50287161   

TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287161(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi:  24nMAssay Description:Binding affinity at Dopamine D3 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287161(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi:  25.1nMAssay Description:Competitive inhibition of [3H]spiperone binding to the human dopamine receptor D3 expressed in CHO cells, expressed as 10log KiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetD(2) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287161(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataKi:  1.89E+3nMAssay Description:Binding affinity at Dopamine D2 receptors in rat striatum by [3H]-spiperone displacement.More data for this Ligand-Target Pair
In DepthDetails Article
TargetD(3) dopamine receptor(Homo sapiens (Human))
TBA

Curated by ChEMBL
LigandPNGBDBM50287161(4-Bromo-1-methoxy-naphthalene-2-carboxylic acid [2...)
Affinity DataEC50:  68nMAssay Description:Compound was evaluated for stimulation of mitogenesis in Dopamine receptor D3 transfected CHO p-5 cellsMore data for this Ligand-Target Pair
In DepthDetails Article