BDBM50318982 2-((1-(3-(9H-carbazol-4-yloxy)-2-hydroxypropyl)piperidin-4-yl)methyl)-5-hydroxy-1H-benzo[de]isoquinoline-1,3(2H)-dione::CHEMBL1084706
SMILES OC(COc1cccc2[nH]c3ccccc3c12)CN1CCC(CN2C(=O)c3cccc4cc(O)cc(C2=O)c34)CC1
InChI Key InChIKey=CLPVTJDKXLZHON-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50318982
Affinity DataKi: 37nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta2 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 250nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta-1 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataKi: 590nMAssay Description:Displacement of [125I]cyanopindolol from human adrenergic beta3 receptor expressed in CHOK1 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 80nMAssay Description:Agonist activity at human adrenergic beta1 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataEC50: 234nMAssay Description:Agonist activity at human adrenergic beta3 receptor expressed in CHOK1 cells assessed as cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair
Affinity DataIC50: 120nMAssay Description:Antagonist activity at human adrenergic beta2 receptor expressed in CHOK1 cells assessed as inhibition of cAMP accumulation by HTRF assayMore data for this Ligand-Target Pair