BDBM50385090 CHEMBL2035603

SMILES Clc1ccccc1-c1nc2c3cc(Br)ccc3oc2c(=O)[nH]1

InChI Key InChIKey=UGRPNQCFWPYERM-UHFFFAOYSA-N

Data  3 IC50

PDB links: 1 PDB ID matches this monomer.

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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50385090   

TargetSerine/threonine-protein kinase pim-2(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50385090(CHEMBL2035603)
Affinity DataIC50:  781nMAssay Description:Inhibition of N-terminal His-tagged human PIM2 expressed in Escherichia coli using AKRRRLSA as substrate after 1 to 2 hrs by luciferasse-luciferin-co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-1(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50385090(CHEMBL2035603)
Affinity DataIC50:  17nMAssay Description:Inhibition of N-terminal His-tagged human PIM1 expressed in Escherichia coli using AKRRRLSA as substrate after 1 to 2 hrs by luciferasse-luciferin-co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSerine/threonine-protein kinase pim-3(Homo sapiens (Human))
Exelixis

Curated by ChEMBL
LigandPNGBDBM50385090(CHEMBL2035603)
Affinity DataIC50:  18nMAssay Description:Inhibition of N-terminal His-tagged human PIM3 expressed in Escherichia coli using AKRRRLSA as substrate after 1 to 2 hrs by luciferasse-luciferin-co...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed