BDBM50414468 CHEMBL1196581::CHEMBL557502
SMILES COc1cccnc1C(=O)N1CCN(CC1)c1ccc(NC(=O)C(C)(C)c2ccccc2)cc1Cl
InChI Key InChIKey=WIHRUDKZTYLJLT-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50414468
Affinity DataKi: 25.1nMAssay Description:Antagonist activity at human NPY Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 25.1nMAssay Description:Antagonist activity at human neuropeptide Y2 receptor in KAN-TS cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: 50.1nMAssay Description:Antagonist activity at rat NPY Y2 receptor expressed in HEK cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: >6.31E+3nMAssay Description:Antagonist activity at human neuropeptide Y1 receptor expressed in CHO cells by [35]GTPgammaS assayMore data for this Ligand-Target Pair
Affinity DataKi: >1.00E+4nMAssay Description:Antagonist activity at human neuropeptide Y5 receptor expressed in HEK293 cells by FLIPR/Ca2+ methodMore data for this Ligand-Target Pair
TargetPotassium voltage-gated channel subfamily H member 2(Homo sapiens (Human))
Glaxosmithkline
Curated by ChEMBL
Glaxosmithkline
Curated by ChEMBL
Affinity DataIC50: 5.01E+4nMAssay Description:Inhibition of human ERGMore data for this Ligand-Target Pair