BDBM50445334 CHEMBL3104247::US9555024, 7

SMILES Fc1ccc(cc1C(=O)NNC(=O)c1cccc(Cl)c1)S(=O)(=O)N1CCOCC1

InChI Key InChIKey=CNZJIFMICCWVNM-UHFFFAOYSA-N

Data  3 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 3 hits for monomerid = 50445334   

TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Utah Research Foundation

US Patent
LigandPNGBDBM50445334(CHEMBL3104247 | US9555024, 7)
Affinity DataIC50: >3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Utah Research Foundation

US Patent
LigandPNGBDBM50445334(CHEMBL3104247 | US9555024, 7)
Affinity DataIC50: >3.00E+3nMAssay Description:The primary assay for compound inhibitory activity was the LSD1 Inhibitor Screening Assay Kit (Cayman Chemical Company, Ann Arbor, Mich.; Cayman Chem...More data for this Ligand-Target Pair
In DepthDetails US Patent
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
University of Utah Research Foundation

US Patent
LigandPNGBDBM50445334(CHEMBL3104247 | US9555024, 7)
Affinity DataIC50: >3.00E+3nMAssay Description:Inhibition of LSD1 (unknown origin) using dimethyl K4 peptide as substrate assessed as resorufin level by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed