BDBM50459262 CHEMBL4213538
SMILES CC(C)[C@H](NC(=O)[C@@H]1CSSC[C@H](NC(=O)[C@H](N)CC(O)=O)C(=O)N[C@@H](Cc2ccc(I)cc2)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)N1)C(O)=O
InChI Key InChIKey=FAZKACLBWZFQSM-RWKAWOQZSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50459262
Affinity DataEC50: 12nMAssay Description:Antagonist activity at UT receptor in Sprague-Dawley rat thoracic aortic ring assessed as reduction in URP-induced contraction by measuring pEC50 for...More data for this Ligand-Target Pair
Affinity DataIC50: <1.00E+3nMAssay Description:Displacement of [Na125I]-synthetic URP from human UT receptor expressed in HEK293 cell membranes incubated for 2 hrs by gamma-countingMore data for this Ligand-Target Pair
Affinity DataEC50: 123nMAssay Description:Agonist activity at human UT receptor expressed in HEK293 cells co-expressing G12-polycistronic BRET biosensor assessed as induction of G12 activatio...More data for this Ligand-Target Pair
Affinity DataEC50: <1.00E+4nMAssay Description:Agonist activity at UT receptor in Sprague-Dawley rat thoracic aortic ring assessed as induction of contractionMore data for this Ligand-Target Pair
Affinity DataEC50: 47nMAssay Description:Agonist activity at human UT receptor expressed in HEK293 cells co-expressing Gq-polycistronic BRET biosensor assessed as induction of Gq activation ...More data for this Ligand-Target Pair
Affinity DataEC50: 1.10nMAssay Description:Antagonist activity at UT receptor in Sprague-Dawley rat thoracic aortic ring assessed as reduction in urotensin-2-induced contraction by measuring p...More data for this Ligand-Target Pair
Affinity DataEC50: 347nMAssay Description:Agonist activity at human UT receptor expressed in HEK293 cells co-expressing beta-arrestin1-polycistronic BRET biosensor assessed as induction of be...More data for this Ligand-Target Pair