BDBM50469449 CHEMBL4277047

SMILES C[C+]1CN(Cc2ccc(CN(C)C)cc12)C(=O)c1cc2cc(Br)ncc2n1C

InChI Key InChIKey=VUJUYQRATLTOLG-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 50469449   

TargetPyroglutamylated RF-amide peptide receptor(Homo sapiens (Human))
Normandy University

Curated by ChEMBL
LigandPNGBDBM50469449(CHEMBL4277047)
Affinity DataIC50:  579nMAssay Description:Antagonist activity at human QRFPR expressed in CHO cells co-expressing Galpha16 assessed as inhibition of 26RFa-induced Ca2+ mobilization preincubat...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed