BDBM50502760 CHEMBL4475503

SMILES C(N1CCN(CC1)[C@H]1CC[C@H](CC1)c1ccccc1)c1cccnc1

InChI Key InChIKey=LKLASWHVKBTLFT-SZPZYZBQSA-N

Data  2 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50502760   

TargetTransient receptor potential cation channel subfamily V member 6(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50502760(CHEMBL4475503)
Affinity DataIC50:  550nMAssay Description:Inhibition of human TRPV6 expressed in HEK293 cells assessed as reduction in Cd2+ influx by calcium-5 fluorescence dye-based FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTransient receptor potential cation channel subfamily V member 6(Homo sapiens (Human))
University Of Bern

Curated by ChEMBL
LigandPNGBDBM50502760(CHEMBL4475503)
Affinity DataIC50:  1.70E+3nMAssay Description:Inhibition of human TRPV6 expressed in HEK293 cells assessed as reduction of Cd2+ influx preincubated for 5 mins followed by CdCl2 addition by calciu...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed