BDBM50521371 CHEMBL4569451

SMILES OC(=O)c1ccc(cc1)-c1cn(nn1)-c1cccnc1

InChI Key InChIKey=CALAFEGXXZJBTB-UHFFFAOYSA-N

Data  4 IC50  1 Kd

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
Find this compound or compounds like it in BindingDB:
   Substructure
Similarity at least:  must be >=0.5
Exact match

Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 5 hits for monomerid = 50521371   

TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521371(CHEMBL4569451)
Affinity DataIC50:  2.00E+4nMAssay Description:Inhibition of fluorescent labelled LBS1 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521371(CHEMBL4569451)
Affinity DataIC50:  1.90E+4nMAssay Description:Inhibition of fluorescent labelled LBS3 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521371(CHEMBL4569451)
Affinity DataIC50:  1.70E+4nMAssay Description:Inhibition of fluorescent labelled LBS2 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521371(CHEMBL4569451)
Affinity DataIC50:  4.26E+5nMAssay Description:Inhibition of 5'-Dy682-labelled LBS1 DNA binding to human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1146...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetORF 73(Human herpesvirus 8)
Institute For Pharmaceutical Research Saarland (Hips)-Helmholtz Centre For Infection Research (Hzi

Curated by ChEMBL
LigandPNGBDBM50521371(CHEMBL4569451)
Affinity DataKd:  2.30E+4nMAssay Description:Binding affinity to human herpesvirus human herpesvirus 8 C-terminal His-tagged LANA oligomerization deficient mutant DBD (1008 to 1146 residues) exp...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed