BDBM50554766 CHEMBL4795492
SMILES CCC(=O)N(Cc1ccccc1)C1(CCN(CCc2ccccc2)CC1)C(=O)NCCc1cccc(F)c1
InChI Key InChIKey=SZQGSEKOXWECKF-UHFFFAOYSA-N
Data 6 EC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 6 hits for monomerid = 50554766
TargetMu-type opioid receptor(Homo sapiens (Human))
St Louis College Of Pharmacy And Washington University
Curated by ChEMBL
St Louis College Of Pharmacy And Washington University
Curated by ChEMBL
Affinity DataEC50: 0.400nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
TargetDelta-type/Mu-type opioid receptor(MOUSE)
St Louis College Of Pharmacy And Washington University
Curated by ChEMBL
St Louis College Of Pharmacy And Washington University
Curated by ChEMBL
Affinity DataEC50: 0.0320nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
St Louis College Of Pharmacy And Washington University
Curated by ChEMBL
St Louis College Of Pharmacy And Washington University
Curated by ChEMBL
Affinity DataEC50: 960nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
TargetMu-type opioid receptor(Homo sapiens (Human))
St Louis College Of Pharmacy And Washington University
Curated by ChEMBL
St Louis College Of Pharmacy And Washington University
Curated by ChEMBL
Affinity DataEC50: 119nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human MOR expressed in human U2OS cell membranes assessed as stimulation beta-arrestin recruitme...More data for this Ligand-Target Pair
TargetDelta-type opioid receptor(Homo sapiens (Human))
St Louis College Of Pharmacy And Washington University
Curated by ChEMBL
St Louis College Of Pharmacy And Washington University
Curated by ChEMBL
Affinity DataEC50: 172nMAssay Description:Agonist activity at EA-fragment beta-arrestin-tagged human DOR expressed in human U2OS cell membranes assessed as stimulation of [35S]-GTPgammaS bind...More data for this Ligand-Target Pair
TargetDelta-type/Mu-type opioid receptor(MOUSE)
St Louis College Of Pharmacy And Washington University
Curated by ChEMBL
St Louis College Of Pharmacy And Washington University
Curated by ChEMBL
Affinity DataEC50: 0.0316nMAssay Description:Agonist activity at MOR/DOR in wild-type C57BL6 mouse spinal cord membranes assessed as stimulation of [35S]-GTPgammaS binding measured after 60 mins...More data for this Ligand-Target Pair