BDBM50558695 CHEMBL4741230
SMILES CC(C)[C@H](NC(=O)[C@@H]1CSSC[C@H](NC(=O)[C@H](CC(O)=O)NC(=O)[C@@H]2CCCN2C(=O)[C@@H](NC(=O)[C@@H](N)CCC(O)=O)[C@@H](C)O)C(=O)N[C@@H](Cc2ccccc2)C(=O)N[C@@H](Cc2c[nH]c3ccccc23)C(=O)N[C@@H](CCCCN)C(=O)N[C@@H](Cc2ccc(O)cc2)C(=O)N1)C(N)=O
InChI Key InChIKey=UFKIKPLPYOYMOM-USJMABIRSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 7 hits for monomerid = 50558695
Affinity DataEC50: 1.5nMAssay Description:Agonist activity at human U-IIR expressed in HEK293-A cells by Fluo4-AM dye based intracellular calcium mobilization assayMore data for this Ligand-Target Pair
Affinity DataIC50: 2nMAssay Description:Displacement of [125I-Tyr9]-U-II from human U-IIR expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand b...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 1(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 1.05E+4nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR1 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 5(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 7.60E+3nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR5 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 3(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 8.64E+3nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR3 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 4(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 1.07E+4nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR4 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair
TargetSomatostatin receptor type 2(Homo sapiens (Human))
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Charit£-Universit£Tsmedizin Berlin
Curated by ChEMBL
Affinity DataIC50: 2.98E+3nMAssay Description:Displacement of [125I-Tyr11]-SS14 from human SSTR2 expressed in HEK293-A cells incubated for 30 mins by gamma counting based competition radioligand ...More data for this Ligand-Target Pair