BDBM50591358 CHEMBL5204703
SMILES Fc1cccc(Cl)c1C1NC(=O)c2c(Cl)cccc2N1
InChI Key InChIKey=LRNRPLFSBRYMGJ-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 5 hits for monomerid = 50591358
Affinity DataIC50: 1.00E+3nMAssay Description:Inhibition of biotinylated histone H3K14 (1 to 20 residues) peptide binding to His6-tagged recombinant human PBRM1 BD2 transfected in Escherichia col...More data for this Ligand-Target Pair
Affinity DataKd: 9.30E+3nMAssay Description:Binding affinity to His-TEV-tagged recombinant human PBRM1 BD2 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM ...More data for this Ligand-Target Pair
TargetTranscription activator BRG1(Homo sapiens (Human))
Medical College Of Wisconsin
Curated by ChEMBL
Medical College Of Wisconsin
Curated by ChEMBL
Affinity DataKd: 6.90E+4nMAssay Description:Binding affinity to N-terminal His-TEV-tagged human SMARCA4 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM by ...More data for this Ligand-Target Pair
TargetProbable global transcription activator SNF2L2(Homo sapiens (Human))
Medical College Of Wisconsin
Curated by ChEMBL
Medical College Of Wisconsin
Curated by ChEMBL
Affinity DataKd: 1.84E+4nMAssay Description:Binding affinity to N-terminal His6-TEV-tagged human SMARCA2B transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM b...More data for this Ligand-Target Pair
Affinity DataKd: 1.01E+4nMAssay Description:Binding affinity to His-TEV-tagged human PBRM1 BD5 transfected in Escherichia coli BL21 (DE3) assessed as dissociation constant at 30 uM by ITC analy...More data for this Ligand-Target Pair