BDBM50596984 CHEMBL5207485
SMILES Fc1cc(F)c(OCc2cccnc2F)c(c1)[C@H]1C[C@@H]1NCC(=O)N1CCC2(CCNC2)CC1
InChI Key InChIKey=AOUYVKAMPAJOPE-NQIIRXRSSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 4 hits for monomerid = 50596984
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Riken Center For Sustainable Resource Science
Curated by ChEMBL
Riken Center For Sustainable Resource Science
Curated by ChEMBL
Affinity DataKi: 80nMAssay Description:Inhibition of human LSD1 assessed as inhibitory constant using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by substrate...More data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] B(Homo sapiens (Human))
Riken Center For Sustainable Resource Science
Curated by ChEMBL
Riken Center For Sustainable Resource Science
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of MAO-B (unknown origin) using tyramine as substrate and measured after 10 mins by peroxidase-coupled reaction methodMore data for this Ligand-Target Pair
TargetAmine oxidase [flavin-containing] A(Homo sapiens (Human))
Riken Center For Sustainable Resource Science
Curated by ChEMBL
Riken Center For Sustainable Resource Science
Curated by ChEMBL
Affinity DataKi: >2.50E+5nMAssay Description:Inhibition of MAO-A (unknown origin) using tyramine as substrate and measured after 10 mins by peroxidase-coupled reaction methodMore data for this Ligand-Target Pair
TargetLysine-specific histone demethylase 1A(Homo sapiens (Human))
Riken Center For Sustainable Resource Science
Curated by ChEMBL
Riken Center For Sustainable Resource Science
Curated by ChEMBL
Affinity DataIC50: 390nMAssay Description:Inhibition of human LSD1 assessed as demethylase activity of LSD1 using Histone H3(1-20)K4me2 peptide as substrate incubated for 10 mins followed by ...More data for this Ligand-Target Pair