BDBM50599557 CHEMBL5196430

SMILES COc1cc2ccn(C\C=C\C(=O)NC3CCCCC3)c(=O)c2cc1OC

InChI Key InChIKey=MEYDDTLLBGAOIV-RMKNXTFCSA-N

Data  2 KI

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 2 hits for monomerid = 50599557   

TargetProteasome subunit beta type-5(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50599557(CHEMBL5196430)
Affinity DataKi:  2.30E+4nMAssay Description:Inhibition of 20S constitutive proteosome beta5c subunit (unknown origin) assessed as substrate hydrolysis using Suc-Leu-Leu-Val-Tyr-AMC as fluorogen...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
University Of Messina

Curated by ChEMBL
LigandPNGBDBM50599557(CHEMBL5196430)
Affinity DataKi:  4.20E+4nMAssay Description:Inhibition of 20S immuno proteosome beta2i subunit (unknown origin) assessed as substrate hydrolysis using Boc-Leu-Arg-Arg-AMC as fluorogenic substra...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed