BDBM518490 US11124509, Compound 63

SMILES Cc1cc(cc(C)c1-c1nc(-c2ccn(C)n2)c([nH]1)-c1ccc2ncsc2c1)C(N)=O

InChI Key InChIKey=VNPFTGHWYKAPNF-UHFFFAOYSA-N

Data  1 IC50

  Tab Delimited (TSV)   2D SDfile   Computed 3D by Vconf -m prep SDfile
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Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB

Found 1 hit for monomerid = 518490   

TargetTGF-beta receptor type-1(Homo sapiens (Human))
Clavius Pharmaceuticals

US Patent
LigandPNGBDBM518490(US11124509, Compound 63)
Affinity DataIC50:  399nMAssay Description:Exemplified compounds were screened in 1% DMSO (final concentration) by 3-fold serial dilutions from 10,000 nM to 0.316 nM to produce an IC50 or at s...More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails US Patent