BDBM639816 US20230391786, Example 285
SMILES Clc1cc(OCC#N)c2c(-c3cn[nH]c3)c3CN(CCn3c2c1Cl)C(=O)[C@@H]1COCCO1
InChI Key
Data 1 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 1 hit for monomerid = 639816
Affinity DataIC50: 12.6nMAssay Description:In vitro inhibition assay of cGAS activity: Add a 5 μL mixture containing 10 mM Tris-Cl pH 7.5, 50 mM NaCl, 5 mM MgCl2, 1 mM DTT, 0.01% Triton X...More data for this Ligand-Target Pair