BDBM82195 Substrate analogue, 13
SMILES CC(=O)OCC(O)=O
InChI Key InChIKey=MLXDUYUQINCFFV-UHFFFAOYSA-N
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 3 hits for monomerid = 82195
Affinity DataKi: 2.45E+7nM ΔG°: -2.28kcal/molepH: 8.1 T: 2°CAssay Description:The PBGS assay is a colorimetric assay based on the reaction between PBG and 4-dimethylaminobenzaldehyde (Ehrlich's reagent). More data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 1.10E+6nMAssay Description:Competitive inhibition of PAM in human DMS53 cells using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair
TargetPeptidyl-glycine alpha-amidating monooxygenase(Homo sapiens (Human))
Australian National University
Curated by ChEMBL
Australian National University
Curated by ChEMBL
Affinity DataIC50: 1.10E+6nMAssay Description:Competitive inhibition of secreted PAM in human DMS53 cell culture medium using as(R)-Tyr-(S)-Val-Gly as substrate after 2 hrs by HPLC analysisMore data for this Ligand-Target Pair