BDBM84799 PF-04764755
SMILES Brc1ccc(cc1)-c1c[nH]c(n1)-c1cc2ccccc2cn1
InChI Key InChIKey=CUBRRNYTHPGDDR-UHFFFAOYSA-N
Data 2 IC50
Activity Spreadsheet -- Enzyme Inhibition Constant Data from BindingDB
Found 2 hits for monomerid = 84799
Affinity DataIC50: 2.95E+3nMpH: 7.5 T: 2°CAssay Description:Inhibition of active p38a MAP kinase by inhibitors was determinedusing a p38a cascade activity assay. A 30-lL reaction mixture wasprepared containing...More data for this Ligand-Target Pair
Affinity DataIC50: 320nMpH: 7.5 T: 2°CAssay Description:Binding of inhibitors to unactivated p38a that leads to decreasedphosphorylation of p38alpha by MKK6 was determined by measuringthe activated p38alph...More data for this Ligand-Target Pair