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Found 54 with Last Name = 'holý' and Initial = 'a'
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50439836(CHEMBL2420072)
Affinity DataKi:  100nMAssay Description:Inhibition of recombinant human HGPRT expressed in Escherichia coli Sphi606 cells by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50304140(9-[2-(1-Phosphonopropan-2-yloxy)ethyl]guanine | CH...)
Affinity DataKi:  100nMAssay Description:Inhibition of human recombinant HGPRT expressed in Escherichia coli by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50304141(9-[2-(1-Phosphonobutan-2-yloxy)ethyl]guanine | CHE...)
Affinity DataKi:  300nMAssay Description:Inhibition of human recombinant HGPRT expressed in Escherichia coli by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50049966(CHEMBL177948 | [4-(2-Amino-6-oxo-1,6-dihydro-purin...)
Affinity DataKi:  400nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360117(CHEMBL1928784)
Affinity DataKi:  500nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50039559(CHEMBL267803 | [5-(2-Amino-6-oxo-1,6-dihydro-purin...)
Affinity DataKi:  500nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293820(2-(2-(2-amino-6-oxo-1,6,7,8-tetrahydropurin-9-yl)e...)
Affinity DataKi:  1.00E+3nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50439833(CHEMBL2420080)
Affinity DataKi:  1.60E+3nMAssay Description:Inhibition of recombinant human HGPRT expressed in Escherichia coli Sphi606 cells by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360122(CHEMBL1928777)
Affinity DataKi:  1.90E+3nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50304138(9-[2-(1-Phosphonopropan-2-yloxy)ethyl]hypoxanthine...)
Affinity DataKi:  2.00E+3nMAssay Description:Inhibition of human recombinant HGPRT expressed in Escherichia coli by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360116(CHEMBL1928783)
Affinity DataKi:  3.00E+3nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360109(CHEMBL1928778)
Affinity DataKi:  3.40E+3nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293821(2-(2-(6-oxo-1,6,7,8-tetrahydropurin-9-yl)ethoxy)et...)
Affinity DataKi:  3.60E+3nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50439834(CHEMBL2420081)
Affinity DataKi:  3.70E+3nMAssay Description:Inhibition of recombinant human HGPRT expressed in Escherichia coli Sphi606 cells by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50361442(CHEMBL1934407)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of human HGPRT by spectrophotometric analysis in absence of PPiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293826((2-(4-oxo-2,3,4,5-tetrahydropyrazolo[3,4-d]pyrimid...)
Affinity DataKi:  4.30E+3nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50439835(CHEMBL2420071)
Affinity DataKi:  4.70E+3nMAssay Description:Inhibition of recombinant human HGPRT expressed in Escherichia coli Sphi606 cells by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50361443(CHEMBL1934409)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of human HGPRT by spectrophotometric analysis in absence of PPiMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50049962(CHEMBL172844 | [7-(2-Amino-6-oxo-1,6-dihydro-purin...)
Affinity DataKi:  5.00E+3nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293819(((2R,3S,4R,5R)-3,4-dihydroxy-5-(6-oxo-1,6,7,8-tetr...)
Affinity DataKi:  5.40E+3nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50439832(CHEMBL2420078)
Affinity DataKi:  5.40E+3nMAssay Description:Inhibition of recombinant human HGPRT expressed in Escherichia coli Sphi606 cells by spectrophotometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293818(((2R,3S,4R,5R)-5-(2-amino-6-oxo-1,6,7,8-tetrahydro...)
Affinity DataKi:  5.80E+3nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293830(CHEMBL561493 | RS-(3-(2-amino-6-oxo-1,6,7,8-tetrah...)
Affinity DataKi:  5.90E+3nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50304139(9-[2-(1-Phosphonobutan-2-yloxy)ethyl]hypoxanthine ...)
Affinity DataKi:  1.00E+4nMAssay Description:Inhibition of human recombinant HGPRT expressed in Escherichia coli by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293835((R)-5-(2-Amino-6-oxo-1,6,7,8-tetrahydro-purin-9-yl...)
Affinity DataKi:  1.23E+4nMpH: 8.5Assay Description:Inhibition of human recombinant HGPRT at pH 8.5 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293831((S)-(1-(5-amino-7-oxo-1,2,6,7-tetrahydro-[1,2,3]tr...)
Affinity DataKi:  1.50E+4nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293835((R)-5-(2-Amino-6-oxo-1,6,7,8-tetrahydro-purin-9-yl...)
Affinity DataKi:  1.90E+4nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360112(CHEMBL19784)
Affinity DataKi:  2.10E+4nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293836(CHEMBL541006 | RS-(1-(2-amino-6-oxo-7,8-dihydro-1H...)
Affinity DataKi:  2.27E+4nMpH: 8.5Assay Description:Inhibition of human recombinant HGPRT at pH 8.5 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360119(CHEMBL1928930)
Affinity DataKi:  2.80E+4nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50225188((2-(2-amino-6-oxo-1,6,7,8-tetrahydropurin-9-yl)eth...)
Affinity DataKi:  2.90E+4nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360114(CHEMBL20283)
Affinity DataKi:  3.10E+4nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293833(((R)-1-(2-amino-8-bromo-6-oxo-1,6,7,8-tetrahydropu...)
Affinity DataKi:  4.10E+4nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50225188((2-(2-amino-6-oxo-1,6,7,8-tetrahydropurin-9-yl)eth...)
Affinity DataKi:  5.59E+4nMpH: 8.5Assay Description:Inhibition of human recombinant HGPRT at pH 8.5 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360115(CHEMBL1928782)
Affinity DataKi:  5.60E+4nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293824((2-(2-amino-8-hydroxy-6-oxo-1,6,7,8-tetrahydropuri...)
Affinity DataKi:  6.80E+4nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360118(CHEMBL1928785)
Affinity DataKi:  7.70E+4nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293834((S)-5-(2-Amino-6-oxo-1,6,7,8-tetrahydro-purin-9-yl...)
Affinity DataKi:  9.00E+4nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50039555(CHEMBL13130 | [5-(6-Oxo-1,6-dihydro-purin-9-yl)-pe...)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360111(CHEMBL1928780)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360121(CHEMBL1928776)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360120(CHEMBL1928931)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360108(CHEMBL1928775)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360110(CHEMBL1928779)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50360113(CHEMBL1928781)
Affinity DataKi: >1.00E+5nMAssay Description:Inhibition of human HGPRTMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293834((S)-5-(2-Amino-6-oxo-1,6,7,8-tetrahydro-purin-9-yl...)
Affinity DataKi:  1.15E+5nMpH: 8.5Assay Description:Inhibition of human recombinant HGPRT at pH 8.5 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293828(CHEMBL560759 | isopropyl(2-(2-amino-6-oxo-1,6,7,8-...)
Affinity DataKi:  1.40E+5nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293823((2-(5-amino-7-oxo-1,2,6,7-tetrahydro-[1,2,3]triazo...)
Affinity DataKi:  1.75E+5nMpH: 7.4Assay Description:Inhibition of human recombinant HGPRT at pH 7.4 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293837((S)-9-[3-hydroxy-2-(phosphonomethoxy)propyl]guanin...)
Affinity DataKi:  1.77E+5nMpH: 8.5Assay Description:Inhibition of human recombinant HGPRT at pH 8.5 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHypoxanthine-guanine phosphoribosyltransferase(Homo sapiens (Human))
Academy Of Sciences Of The Czech Republic

Curated by ChEMBL
LigandPNGBDBM50293838((2-(6-oxo-1,6,7,8-tetrahydropurin-9-yl)ethoxy)meth...)
Affinity DataKi:  1.82E+5nMpH: 8.5Assay Description:Inhibition of human recombinant HGPRT at pH 8.5 by spectrophotometric assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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