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Found 37 with Last Name = 'koshino' and Initial = 'h'
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataKi:  4.00E+3nMAssay Description:Inhibition of wild type human USP5 expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate after 60 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataKi:  1.25E+4nMAssay Description:Competitive inhibition of wild type human USP5 expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrateMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50145539((2S,4R)-2,4-Dihydroxy-6-[2-[(R)-1-((R)-5-hydroxy-1...)
Affinity DataIC50:  0.5nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50145538((S)-1-Benzyl-5-((R)-2-{(R)-4-[2-[(3S,5R)-3,5-dihyd...)
Affinity DataIC50:  1.90nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50145540((S)-5-((R)-2-{(R)-4-[2-[(3S,5R)-3,5-Dihydroxy-2-me...)
Affinity DataIC50:  10nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50089194((R)-N*4*-Hydroxy-N*1*-[(S)-1-((S)-2-hydroxymethyl-...)
Affinity DataIC50:  20nMAssay Description:Inhibition of Staphylococcus aureus peptide deformylase using N-formylmethionine-alanine-serine as substrate by spectrophotometryMore data for this Ligand-Target Pair
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50404242(CHEMBL2114211)
Affinity DataIC50:  30nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50404243(CHEMBL2114212 | CHEMBL3350688)
Affinity DataIC50:  50nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetVitamin D3 receptor(Gallus gallus)
University Of Tokyo

Curated by ChEMBL
LigandPNGBDBM50223417(CHEMBL3350292)
Affinity DataIC50: >100nMAssay Description:In vitro relative binding affinity for chick intestinal vitamin D3 receptor compared to [3H]-1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl oligopeptidase family protein(Flavobacterium psychrophilum (strain JIP02/86 / AT...)
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50455076(CHEMBL4214751)
Affinity DataIC50:  770nMAssay Description:Inhibition of Flavobacterium POP preincubated for 5 mins followed by Z-Gly-Pro-pNA substrate measured after 30 minsMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50455075(CHEMBL4209844)
Affinity DataIC50:  950nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetProlyl oligopeptidase family protein(Flavobacterium psychrophilum (strain JIP02/86 / AT...)
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50269566(CHEMBL458248 | polyozellin)
Affinity DataIC50:  1.20E+3nMAssay Description:Inhibition of Flavobacterium POP preincubated for 5 mins followed by Z-Gly-Pro-pNA substrate measured after 30 minsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50269567(CHEMBL515528 | Kynapcin-12)
Affinity DataIC50:  1.25E+3nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50046279(CHEMBL3314376)
Affinity DataIC50:  1.40E+3nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 4(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  1.50E+3nMAssay Description:Inhibition of human USP4 using Ub-AMC as substrate after 60 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50269566(CHEMBL458248 | polyozellin)
Affinity DataIC50:  2.72E+3nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437695(CHEMBL1923233)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of USP5 in human Z138 cells after 1 hr by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProbable ubiquitin carboxyl-terminal hydrolase FAF-X(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437695(CHEMBL1923233)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of USP9x in human Z138 cells after 1 hr by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase isozyme L1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437695(CHEMBL1923233)
Affinity DataIC50:  3.00E+3nMAssay Description:Inhibition of UCH-L1 in human Z138 cells after 1 hr by immunoblotting analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50046278(CHEMBL3314375)
Affinity DataIC50:  3.50E+3nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase 14(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437694(CHEMBL1410015)
Affinity DataIC50:  4.00E+3nMAssay Description:Inhibition of human USP14More data for this Ligand-Target Pair
TargetUbiquitin carboxyl-terminal hydrolase 5(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  5.90E+3nMAssay Description:Inhibition of wild type human USP5 expressed in Escherichia coli BL21(DE3) using Ub-AMC as substrate after 60 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50046273(CHEMBL3314370)
Affinity DataIC50:  1.15E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50046275(CHEMBL3314372)
Affinity DataIC50:  1.49E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50046276(CHEMBL3314373)
Affinity DataIC50:  1.51E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50046188(CHEMBL3238007)
Affinity DataIC50:  1.52E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-1(Homo sapiens (Human))
Hirosaki University

Curated by ChEMBL
LigandPNGBDBM50270495(CHEMBL4126890)
Affinity DataIC50:  1.73E+4nMAssay Description:Inhibition of human erythrocyte 20s proteasome caspase-like activity using Z-LLE-MCA as substrate pretreated for 10 mins followed by substrate additi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50046277(CHEMBL3314374)
Affinity DataIC50:  1.77E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-5(Homo sapiens (Human))
Hirosaki University

Curated by ChEMBL
LigandPNGBDBM50270495(CHEMBL4126890)
Affinity DataIC50:  1.85E+4nMAssay Description:Inhibition of human erythrocyte 20s proteasome chymotrypsin-like activity using Suc-LLVY-MCA as substrate pretreated for 10 mins followed by substrat...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetUbiquitin carboxyl-terminal hydrolase isozyme L1(Homo sapiens (Human))
Tokyo University Of Agriculture

Curated by ChEMBL
LigandPNGBDBM50437693(VIALININ A)
Affinity DataIC50:  2.23E+4nMAssay Description:Inhibition of human UCH-L1 using Ub-AMC as substrate after 60 mins by fluorometric analysisMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50379509(CHEMBL2012550)
Affinity DataIC50:  3.58E+4nMAssay Description:Inhibition of Staphylococcus aureus peptide deformylase using N-formylmethionine-alanine-serine as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProteasome subunit beta type-2(Homo sapiens (Human))
Hirosaki University

Curated by ChEMBL
LigandPNGBDBM50270495(CHEMBL4126890)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of human erythrocyte 20s proteasome trypsin-like activity using Boc-LRR-MCA as substrate pretreated for 10 mins followed by substrate addi...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50046272(CHEMBL3314369)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50046263(CHEMBL3314368)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Homo sapiens (Human))
Riken Csrs

Curated by ChEMBL
LigandPNGBDBM50046274(CHEMBL3314371)
Affinity DataIC50: >5.00E+4nMAssay Description:Inhibition of prolyl oligopeptidase (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeptide deformylase(Staphylococcus aureus)
Korea Research Institute Of Bioscience And Biotechnology

Curated by ChEMBL
LigandPNGBDBM50379510(CHEMBL2012551)
Affinity DataIC50:  1.00E+5nMAssay Description:Inhibition of Staphylococcus aureus peptide deformylase using N-formylmethionine-alanine-serine as substrate by spectrophotometryMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlycogen synthase kinase-3 beta(Homo sapiens (Human))
Iwate University

Curated by ChEMBL
LigandPNGBDBM50465052(CHEMBL4288015)
Affinity DataIC50:  1.78E+5nMAssay Description:Inhibition of human GSK-3beta using peptide substrateMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed